Arimidex benefits and other things
As you know, anabolic steroids are potent substances that cause muscle hypertrophy. Their effects are currently being actively studied both in medicine and in the field of sports. And the first thing i want to say, that safe steroids do not exist. Every steroids group has its own couple of side effects. And, to avoid aromatization associated effects, we use some drugs, called aromatase inhibitors. At this blog section we will talk about one of that drug – Arimidex.
What is Arimidex?
Arimidex is a medicine that was originally created to treat breast tumors in women. This drug reduce estrogen receptors in problem areas. As an antiestrogen drug Arimidex available in tablet form. However, today we practically do not use this drug in medical practice. In the future, for the ability to reduce estrogen, it began to be used in sports with the use of anabolic steroids. As you know, using of steroids raise the level of estrogen in the blood.
The drug was synthesized at the end of the 20th century and literally for 20 years to be in the medicine cabinet of athletes around the world. But the main consumers of this drug are bodybuilders and athletes of heavy sports. Arimidex helps to avoid gynecomastia, that is, growth of the mammary glands, eliminates edema and other negative side effects that often accompany the anabolics courses. It is also reduce water retention in the body, which leads to a decrease in pressure and a number of other positive aspects.
Athelets use Arimidex to counter the increased level of female sex hormones. This is observed against the background of an increase in testosterone and gonadotropin levels. This often happens when athletes and bodybuilders take special medications to increase muscle mass, increase stamina and physical strength, and develop beautifully outlined muscles.
As you know, Arimidex belong to aromatase inhibitors group. So, what about a goal of taking that drugs in sport?
Aromatase inhibitors or blockers is a class of drugs that are used to lower blood estrogen concentrations and increase levels of testosterone and gonadotropin hormones. Aromatase blockers are also used to treat and prevent gynecomastia in men.
In bodybuilding, aromatase inhibitors are most often used during a course of anabolic steroids for:
- gynecomastia prevention
- increased levels of anabolic hormones in the blood
- increased relief (by eliminating the negative effects of estrogen)
- hypertension prevention
- decrease in estrogenic suppression of the axis of the hypothalamus-pituitary-testes, which leads to a faster recovery.
When you build a course, you should remember that not all anabolic steroids are subject to aromatization. The use is justified with the introduction of drugs such as testosterone and its derivatives. Slightly aromatized boldenone and halotestin.
Few words about effects
Arimidex has pronounced effects: only one milligram of the active substance can lower the content of estradiol in the blood by 80%! Even Tamoxifen, quite popular with bodybuilders, cannot be compared with Anastrozole in terms of its effect. However, the drugs have a different principle of action, so the comparison between them is unlikely to be correct.
There’re some effects of Arimidex use:
- Potent aromatase inhibitor;
- Reduces operatively the level of estradiol;
- Reduces water retention in the body;
- The rapid inclusion in the work of the active substance, after 2-3 hours, the concentration of estrogen decreases;
- Improves muscle stiffness and quality.
One of the most important properties of the drug is a fairly quick effect. The maximum concentration of the active substance observe in the blood after a couple of hours after injection. In this case, the suppression of the aromatization process occurs as soon as possible. Therefore, Arimidex is one of the most effective drugs for athletes who have a tendency to aromatize.
When to take Arimidex?
Most athletes are reduce to use of aromatase inhibitors when the first signs of gynecomastia appear (swelling, itching in the nipple, redness). However, this approach is not optimal.
The most rational solution is to perform an estradiol test after about 10 days of taking anabolic steroids with short half-lives (testosterone propionate, methandrostenolone) or after 3-4 weeks of administration of long esters (enanthate, sustanon, cypionate). Then you can take an average dosage of Arimidex of 0.5 mg every other day. After 10 days you must perform a control analysis of estradiol and the correct the dosage according to the results.
A compromise option is to use a moderate or low dosage of Arimidex with an orientation to subjective sensations. If after the appointment there is a drop in libido, erectile dysfunction, depression, then it is necessary to lower the dose.
So what about Arimidex dosage, and how to take it?
Arimidex is a potent substance. Therefore, you should use it either under the supervision of doctors or experienced athletes and the mandatory delivery of tests.
Since the drug is short-acting, you can take Arimidex every other day or every day. It is depending due to analysis and condition of the athlete.
You need to start taking the drug only if necessary and at the first signs of gynecomastia (itching and pain in the nipples, large swelling). Usually start with dosages of 0.25 mg once a day and increase to 1 mg.
The duration of the course of taking Arimidex should not exceed three weeks, otherwise there is a likelihood of a decrease in estrogen to too low an indication.
In order for the active substance to enter the bloodstream as soon as possible, Anastrozole should be taken before meals, washed down with a large volume of water.
We are do not recommend using of Arimidex by women. Becouse of its negative effect on the hormonal system of this gender. Hormonal changes are possible, which will be difficult to restore.
Did you think that there are no side effects?
Like any medicine, Arimidex has side effects. They mainly manifest themselves in people with individual intolerance to the active substance.
Side effects from the drug are relatively rare. As a rule, they are associated with intolerance to the active ingredients or exceeding the recommended dosage.
There are most common Arimidex side effects:
- rapid fatigue
- redness of the skin
- various negative manifestations of the gastrointestinal tract.
You should discard Arimidex in case of chronic diseases of the cardiovascular system. This is due to the fact that the drug actively counteracts the side effects of taking steroids, but at the same time it blocks the production of “good” cholesterol, which can lead to heart problems. For this reason, athletes who have diseases of the cardiovascular system should consult a doctor before taking Anastrozole or prefer drugs with a similar effect, but with a different mechanism of action on the body.
Arimidex vs Aromasin: let’s the battle begin!
What medicines are aromatase inhibitors that are effective in sports practice? The list is actually not very large. “Classical” drugs of this type include: letrozole (Femara drug and others), exemestane (Aromasin and others) and anastrozole (Arimidex and others). These are the most popular and common blockers, the effectiveness of which is not in doubt (proven in many studies). Two of them, Arimidex and Aromasin are most popular aromatase blockers among athelets. You already know, why Arimidex is one of them. So let’s talk about other one – Aromasin.
So, exemestane is a fairly popular aromatase inhibitor, in structure most similar to the steroid hormone androstenedione. It does not have estrogenic or progestogen activity. In fact, when you take, even in high doses, only antiestrogenic and insignificant androgenic activity are possible. However, it does not affect the biosynthesis of aldosterone and cortisol in the adrenal glands.
The main difference between Aromasin and Arimidex that when you take first one, a slight increase in serum FSH and LH hormones is possible (even when using low dosages). This useful effect most likely develops according to the feedback principle (a decrease in estrogen content leads to an increase in the secretion of gonadotropins in the pituitary gland).
A short afterword: Arimidex like the other inhibitos described before, you can order in our store theroids.ws. And the fact that you can quickly and easily order anastrozole in our store. If you are faced with the need for its application, then feel free to go to our website and buy. Favorable price, discounts, convenient service and delivery, reliability – all this you will find. Also on the virtual shelves of our store you will find many other drugs that are popular and effective in sports practice, ranging from steroids and peptides to hormone growth drugs.